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Image Search Results
Journal: Molecules
Article Title: SAR by Space: Enriching Hit Sets from the Chemical Space
doi: 10.3390/molecules24173096
Figure Lengend Snippet: Investigational drugs—bromodomain 4 (BRD4) inhibitors.
Article Snippet: All TR-FRET assays and IC 50 measurements were performed using
Techniques:
Journal: Molecules
Article Title: SAR by Space: Enriching Hit Sets from the Chemical Space
doi: 10.3390/molecules24173096
Figure Lengend Snippet: Known BRD4 inhibitors—analogs of the series identified in this work.
Article Snippet: All TR-FRET assays and IC 50 measurements were performed using
Techniques:
Journal: Molecules
Article Title: SAR by Space: Enriching Hit Sets from the Chemical Space
doi: 10.3390/molecules24173096
Figure Lengend Snippet: Most active BRD4 inhibitors identified after TR-FRET (time-resolved fluorescence energy transfer) assay.
Article Snippet: All TR-FRET assays and IC 50 measurements were performed using
Techniques: Fluorescence
Journal: Marine Drugs
Article Title: Inhibitors of BRD4 Protein from a Marine-Derived Fungus Alternaria sp. NH-F6
doi: 10.3390/md15030076
Figure Lengend Snippet: Inhibition rates of compounds 1 – 24 against BRD4 protein a .
Article Snippet:
Techniques: Inhibition